Impact of Target Warhead and Linkage Vector on Inducing Protein Degradation: Comparison of Bromodomain and Extra-Terminal (BET) Degraders Derived from Triazolodiazepine (JQ1) and Tetrahydroquinoline (I-BET726) BET Inhibitor Scaffolds. (2018)
Attributed to:
A Systems Approach for the Fragment-Based Development of Selective Chemical Probes of Bromodomain Function
funded by
BBSRC
Abstract
No abstract provided
Bibliographic Information
Digital Object Identifier: http://dx.doi.org/10.1021/acs.jmedchem.6b01912
PubMed Identifier: 28595007
Publication URI: http://europepmc.org/abstract/MED/28595007
Type: Journal Article/Review
Volume: 61
Parent Publication: Journal of medicinal chemistry
Issue: 2
ISSN: 0022-2623