Stereochemical inversion at a 1,4-cyclohexyl PROTAC linker fine-tunes conformation and binding affinity. (2024)
Abstract
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Bibliographic Information
Digital Object Identifier: http://dx.doi.org/10.1016/j.bmcl.2024.129861
PubMed Identifier: 38942127
Publication URI: http://europepmc.org/abstract/MED/38942127
Type: Journal Article/Review
Volume: 110
Parent Publication: Bioorganic & medicinal chemistry letters
ISSN: 0960-894X